1: With calcium carbonate in chloroform; water Addition; 16 h; 2: With ammonia in methanol T=0°C; Substitution; 3 h;
参考文献
Ulhaq, Saraj; Chinje, Edwin C.; Naylor, Matthew A.; Jaffar, Mohammed; Stratford, Ian J.; Threadgill, Michael D.
Bioorganic and Medicinal Chemistry, 1999 , vol. 7, # 9 p. 1787 - 1796