反应条件
1: 80 percent / acetic acid / 1.) 42 h, 28 deg C, 2.) 5 h, 50 deg C 2: 78 percent / various solvent(s) / 3 h / 190 - 195 °C 3: 93 percent / H2 / 5 percent Pd/C / ethyl acetate / 1 h / 40 °C View Scheme
参考文献
Boltze; Brendler; Jacobi; Opitz; Raddatz; Seidel; Vollbrecht
Arzneimittel-Forschung/Drug Research, 1980 , vol. 30, # 8 A p. 1314 - 1325