(3-溴苯基)(环丙基)甲胺合成路线 (共 1 条)
反应条件
1: in tetrahydrofuran; methanol
T=0 - 50°C; 4 h;
2: With sodium tetrahydroborate in tetrahydrofuran; methanol
T=0°C; 2.5 h;
3: With water; ammonium chloride in tetrahydrofuran; methanol
参考文献
ASTRAZENECA AB; ASTEX THERAPEUTICS LTD
Patent: WO2008/63114 A1, 2008 ;
Location in patent: Page/Page column 35-36 ;
WO 2008/063114 A1