反应条件
1: 42 percent / 28-30percent NH3 / H2O / 16 h / 150 °C / 36200.4 Torr 2: 86 percent / LiAlH4 / tetrahydrofuran / 1.) 5 h, reflux, 2.) 36 h, r.t. View Scheme
参考文献
Low, Eddy; Kim, Bum; Francavilla, Charles; Shiau, Timothy P.; Turtle, Eric D.; O'Mahony, Donogh J.R.; Alvarez, Nichole; Houchin, Ashley; Xu, Ping; Zuck, Meghan; Celeri, Chris; Anderson, Mark B.; Najafi, Ramin; Jain, Rakesh K.
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 12 p. 3682 - 3685