1: 2-(nitromethylene)tetrahydropyrimidine With sodium hydride in N,N-dimethyl-formamide; mineral oil
T=0 - 5°C; 0.666667 h;
2: 1-iodo-butane in N,N-dimethyl-formamide; mineral oil
T=20°C;
参考文献
Kalisiak, Jaroslaw; Ralph, Erik C.; Cashman, John R.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 1 p. 465 - 474
Emschwiller
Comptes Rendus Hebdomadaires des Seances de l'Academie des Sciences, 1931 , vol. 192, p. 800,800 Anm.
Annales de Chimie (Cachan, France), 1932 , vol. <10>17, p. 425