N-(2-氨基甲酰-3-甲氧基苯基)草氨酸乙酯合成路线 (共 5 条)
反应条件
pyridine in dichloromethane
参考文献
Sellstedt; Guinosso; Begany; Bell; Rosenthale
Journal of Medicinal Chemistry, 1975 , vol. 18, # 9 p. 926 - 933
反应条件
1: TsNH2, PCl5 / 185 - 187 °C
2: methanol
3: aq. N2H4 / Raney-Ni / ethanol
4: Py / CH2Cl2
View Scheme
参考文献
Sellstedt; Guinosso; Begany; Bell; Rosenthale
Journal of Medicinal Chemistry, 1975 , vol. 18, # 9 p. 926 - 933
反应条件
1: aq. N2H4 / Raney-Ni / ethanol
2: Py / CH2Cl2
View Scheme
参考文献
Sellstedt; Guinosso; Begany; Bell; Rosenthale
Journal of Medicinal Chemistry, 1975 , vol. 18, # 9 p. 926 - 933
反应条件
1: methanol
2: aq. N2H4 / Raney-Ni / ethanol
3: Py / CH2Cl2
View Scheme
参考文献
Sellstedt; Guinosso; Begany; Bell; Rosenthale
Journal of Medicinal Chemistry, 1975 , vol. 18, # 9 p. 926 - 933
参考文献
American Home Products Corporation
Patent: US4137325 A1, 1979 ;