反应条件
1: (i) Mg, Et2O, (ii) /BRN= 1633582/
2: (i) NaBH4, NaOH, EtOH, (ii) /BRN= 385737/
3: (i) NaH, benzene, DMF, (ii) /BRN= 2042818/, KI, (iii) TsOH, toluene
View Scheme
参考文献
Bicking; Robb; Smith; Cragoe Jr.
Journal of Medicinal Chemistry, 1977 , vol. 20, # 1 p. 35 - 43