反应条件
1: tert-butyl alcohol
2: n-butyllithium; N,N,N',N,-tetramethylethylenediamine
3: N,N-dimethyl-formamide; methanol; dichloromethane
View Scheme
参考文献
ABBVIE INC.; Vasudevan, Anil; Penning, Thomas Dale; Chen, Huanming; Liang, Bo; Wang, Shaohui; Zhao, Zhongqiang; Chai, Dikun; Yang, Leifu; Gao, Yingxiang; Pliushchev, Marina
Patent: US2014/171429 A1, 2014 ;