1: With N,N-dibenzyl-O-benzyl-L-α-aspartyl-L-proline methyl ester in toluene T=0 - 20°C; 48 h; Inert atmosphere; 2: With hydrogenchloride in water; toluene Inert atmosphere; optical yield given as percent eeenantioselective reaction;
参考文献
Kang, Seock Yong; Park, Yong Sun
European Journal of Organic Chemistry, 2012 , # 9 p. 1703 - 1706
1: With chiral Cu(BozPHOS)2OTf; P(O)(NH2)PPh2 in toluene T=25°C; 48 h; 2: With hydrogenchloride in toluene 8 h; Title compound not separated from byproducts;
参考文献
Cote, Alexandre; Charette, Andre B.
Journal of Organic Chemistry, 2005 , vol. 70, # 26 p. 10864 - 10867
