(9CI)-1-(氰基乙酰基)-1,2,3,4-四氢-喹啉合成路线 (共 1 条)
反应条件
benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide
T=0 - 25°C; 14 - 18 h;
参考文献
CADILA HEALTHCARE LIMITED
Patent: WO2009/87649 A1, 2009 ;
Location in patent: Page/Page column 28-29 ;
WO 2009/087649 A1