反应条件
1: 69 percent / ethyl nitrite, HCl / ethanol / 2 h / 35 °C
2: 65 percent / conc.HCl, H2 / 10percent Pd/C / ethanol / Ambient temperature
View Scheme
参考文献
Perrone; Berardi; Bettoni; Tortorella; Cuomo; Racagni; Juliano; Rovescalli
European Journal of Medicinal Chemistry, 1987 , vol. 22, # 5 p. 417 - 419