1-乙酰基-4-(2-氯乙基)哌嗪合成路线 (共 2 条)
反应条件
thionyl chloride in chloroform T=0°C; 1.83333 h; Heating / reflux;
参考文献
PFIZER LIMITED; PFIZER INC.
Patent: WO2005/82866 A2, 2005 ;
Location in patent: Page/Page column 100 ;
WO 2005/082866 A2
反应条件
potassium iodide; sodium carbonate in 3-methyl-butan-2-one; dichloromethane; water