1: With nitric acid in water; acetic acid
T=10 - 20°C; 18 h;
2: With sodium hydroxide; water in acetic acid
T=15 - 50°C; 21 h;
3: With hydrogenchloride in water; acetic acid
pH=~ 8;
参考文献
ALTANA PHARMA AG
Patent: WO2007/12650 A1, 2007 ;
Location in patent: Page/Page column 27-28 ;