[4-(2-吡嗪基)苯基]甲醇合成路线 (共 1 条)
反应条件
potassium phosphate; tetrakis(triphenylphosphine) palladium(0) in 1,4-dioxane; water
T=80°C; Inert atmosphere;
参考文献
ARENA PHARMACEUTICALS, INC.; JONES, Robert M.; BUZARD, DAniel J.; HAN, Sangdon; KIM, Sun He; LEHMANN, Juerg; ULLMAN, Brett; MOODY, Jeanne V.; ZHU, Xiuwen; STIRN, Scott
Patent: WO2010/11316 A1, 2010 ;
Location in patent: Page/Page column 76-77 ;
WO 2010/011316 A1