1-(苯甲酰基氧基)-1H-1,2,3-苯并噻唑合成路线 (共 31 条)
反应条件
triethylamine; benzoic acid in dichloromethane
参考文献
Fujisawa Pharmaceutical Co., Ltd.
Patent: US4242507 A1, 1980 ;
反应条件
triethylamine; benzoic acid in chloroform
参考文献
Fujisawa Pharmaceutical Co., Ltd.
Patent: US4242507 A1, 1980 ;
反应条件
pyridine in various solvent(s)
1 h; Ambient temperature;
参考文献
Ueda, Mitsuru; Oikawa, Hideaki; Teshirogi, Takuma
Synthesis, 1983 , # 11 p. 908 - 909
反应条件
triethylamine in acetonitrile
12 h; Ambient temperature;
参考文献
Topuzyan, V. O.; Martirosyan, M. S.
Journal of Organic Chemistry USSR (English Translation), 1991 , vol. 27, # 11.2 p. 2148 - 2153
Zhurnal Organicheskoi Khimii, 1991 , vol. 27, # 11 p. 2418 - 2424
反应条件
in water; acetonitrile
T=20°C; Flow reactor;
参考文献
Nagaki, Aiichiro; Takahashi, Yusuke; Yoshida, Jun-Ichi
Chemistry - A European Journal, 2014 , vol. 20, # 26 p. 7931 - 7934
反应条件
N-ethyl-N,N-diisopropylamine in tetrahydrofuran
T=0°C;
参考文献
Vasantha; Sureshbabu, Vommina V.
Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry, 2010 , vol. 49, # 6 p. 812 - 817
反应条件
in acetone
4 h; Heating;
参考文献
Katritzky, Alan R.; Malhotra, N.; Fan, Wei-Quiang; Anders, Ernst
Journal of the Chemical Society, Perkin Transactions 2: Physical Organic Chemistry (1972-1999), 1991 , # 10 p. 1545 - 1547
反应条件
1: 70 percent / benzene / 2 h / Heating
2: 80 percent / pyridine / various solvent(s) / 1 h / Ambient temperature
View Scheme
参考文献
Ueda, Mitsuru; Oikawa, Hideaki; Teshirogi, Takuma
Synthesis, 1983 , # 11 p. 908 - 909
反应条件
1.1: n-butyllithium / tetrahydrofuran; hexane / 0 h / -20 °C / |Flow reactor
1.2: -20 °C / |Flow reactor
2.1: acetonitrile; water / 20 °C / |Flow reactor
View Scheme
参考文献
Nagaki, Aiichiro; Takahashi, Yusuke; Yoshida, Jun-Ichi
Chemistry - A European Journal, 2014 , vol. 20, # 26 p. 7931 - 7934
反应条件
1: tetrahydrofuran / 0.02 h / 78 °C
2: acetonitrile; water / 20 °C / |Flow reactor
View Scheme
参考文献
Nagaki, Aiichiro; Takahashi, Yusuke; Yoshida, Jun-Ichi
Chemistry - A European Journal, 2014 , vol. 20, # 26 p. 7931 - 7934