反应条件
1: 4-Hydroxy-naphthalene-1-carbaldehyde With sodium hydride in tetrahydrofuran; N,N-dimethyl-formamide
T=0°C; 0.5 h;
2: 1-iodo-propane in tetrahydrofuran; N,N-dimethyl-formamide
T=20°C; 2 h;
参考文献
Daiichi Sankyo Company, Limited
Patent: EP1914229 A1, 2008 ;
Location in patent: Page/Page column 109 ;