反应条件
1: sodium hydroxide / N,N-dimethyl-formamide / 3 h / 20 °C
2: hydrogenchloride / 1,4-dioxane / 12 h / 20 °C / |Cooling with ice
View Scheme
参考文献
Mooring, Suazette Reid; Liu, Jin; Liang, Zhongxing; Ahn, Jeffrey; Hong, Samuel; Yoon, Younghyoun; Snyder, James P.; Shim, Hyunsuk
ChemMedChem, 2013 , vol. 8, # 4 p. 622 - 632