5-氨基-6-氯-1H-嘧啶-4-硫酮合成路线 (共 3 条)
参考文献
Yadrovskaya, V.; Nemeryuk, M. P.; Safonova, T. S.
Pharmaceutical Chemistry Journal, 1989 , vol. 23, # 6 p. 518 - 521
Khimiko-Farmatsevticheskii Zhurnal, 1989 , vol. 23, # 6 p. 730 - 733
反应条件
ammonia; water; nickel in ethanol T=20 - 80°C;
参考文献
ELAN PHARMACEUTICALS, INC.
Patent: WO2007/8563 A2, 2007 ;
Location in patent: Page/Page column 88 ;
参考文献
BIOCRYST PHARMACEUTICALS, INC.; BABU, Yarlagadda, S.; CHAND, Pooran; KOTIAN, Pravin, L.; KUMAR, V., Satish
Patent: WO2010/14930 A2, 2010 ;
Location in patent: Page/Page column 50 ;
WO 2010/014930 A2