1: With sodium hydride in N,N-dimethyl-formamide; acetonitrile T=0°C; 2 h; 2: With cis amino chloride in N,N-dimethyl-formamide; acetonitrile T=0°C; 5 h; Further stages.;
参考文献
Wang; Guziec Jr.
Journal of Organic Chemistry, 2001 , vol. 66, # 25 p. 8293 - 8296