1: With oxalyl dichloride; dimethyl sulfoxide in dichloromethane T=-78°C; 2: With triethylamine in monofluorodichloromethane T=-78 - 0°C; 0.666667 h;
参考文献
De Almeida, Gabriela; Sletten, Ellen M.; Nakamura, Hitomi; Palaniappan, Krishnan K.; Bertozzi, Carolyn R.
Angewandte Chemie - International Edition, 2012 , vol. 51, # 10 p. 2443 - 2447