反应条件
potassium carbonate in N,N-dimethyl-formamide
1.) 0 deg C, 30 min, 2.) RT, 24 h;
参考文献
Guo, Hui-Fang; Shao, Hua-Yi; Yang, Zhao-Yong; Xue, Si-Tu; Li, Xue; Liu, Zong-Ying; He, Xiao-Bo; Jiang, Jian-Dong; Zhang, Yue-Qin; Si, Shu-Yi; Li, Zhuo-Rong
Journal of Medicinal Chemistry, 2010 , vol. 53, # 4 p. 1819 - 1829