反应条件
1: 1.) 1.1-carbonyldiimidazole / 1.) THF, RT, 1 h, 2.) THF, RT, 24 h
2: 95 percent / aq. LiOH / dioxane / 24 h
View Scheme
参考文献
Padia, Janak K.; Field, Mark; Hinton, Joanna; Meecham, Ken; Pablo, Julius; Pinnock, Rob; Roth, Bruce D.; Singh, Lakhbir; Suman-Chauhan, Nirmala; Trivedi, Bharat K.; Webdale, Louise
Journal of Medicinal Chemistry, 1998 , vol. 41, # 7 p. 1042 - 1049