反应条件
1: 1.) tritone B / 1.) DMF; 2.) DMF, 5 h 2: 80 percent / HONB, DCCI / dimethylformamide / 1.) 2 h, -20 deg C; 2.) 3 h, room temperature 3: 98 percent / HCl, CH3COOH, C2H5SH / 0.75 h / Ambient temperature 4: 86 percent / N-methylmorpholine / 48 h View Scheme
参考文献
Pharmazie, , vol. 43, # 1 p. 10 - 11