反应条件
1: 1) BCl3, 2) Ag2CO3 / 1) CH2Cl2, -50 deg C to r.t., 2.5 h, 2) 20 min 2: H2O / methanol / 48 °C / pH 8.5 (phosphate or carbonate buffer) View Scheme
参考文献
Atkinson, Jeffrey; Morand, Peter; Arnason, John T.; Niemeyer, Hermann M.; Bravo, Hector R.
Journal of Organic Chemistry, 1991 , vol. 56, # 5 p. 1788 - 1800