5-甲氧基-6-甲基-2,1,3-苯并恶二唑合成路线 (共 2 条)
反应条件
phosphorous acid trimethyl ester in ethanol
1 h; Heating / reflux;
参考文献
Active Biotech AB
Patent: US2005/192289 A1, 2005 ;
Location in patent: Page/Page column 9 ;
反应条件
1: NaOCl
2: NH2OH
View Scheme
参考文献
Angeloni,A.S. et al.
Tetrahedron, 1974 , vol. 30, p. 3849 - 3857