1: [3H]-L-Alanine With lithium aluminium tetrahydride in tetrahydrofuran T=0°C; Heating / reflux; 2: With sodium hydroxide in tetrahydrofuran; water T=20°C; 3 h; 3: benzyl chloroformate With sodium hydroxide in tetrahydrofuran; water 1 h;
参考文献
JERINI AG
Patent: WO2009/36996 A2, 2009 ;
Location in patent: Page/Page column 99-100 ;
WO 2009/036996 A2