反应条件
1: 90 percent
2: 60 percent / dicyclohexylcarbodiimide / ethyl acetate / 1.) 1 h, 0 deg C, 2.) 24 h, r.t.
View Scheme
参考文献
Napolitano, Roberta; Pariani, Giorgio; Fedeli, Franco; Baranyai, Zsolt; Aswendt, Markus; Aime, Silvio; Gianolio, Eliana
Journal of Medicinal Chemistry, 2013 , vol. 56, # 6 p. 2466 - 2477