1: 2-amino-3-chloro-1,4-dihydro-1,4-dioxonaphthalene With tetrakis(triphenylphosphine) palladium(0); potassium carbonate in tetrahydrofuran; water
T=20°C; 0.5 h;
2: 3,4,5-trimethoxyphenylboronic acid in tetrahydrofuran; water
T=20°C; Suzuki coupling; Reflux;
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Kyle Hadden; Hill, Stephanie A.; Davenport, Jason; Matts, Robert L.; Blagg, Brian S.J.
Bioorganic and Medicinal Chemistry, 2009 , vol. 17, # 2 p. 634 - 640
Zincke
Justus Liebigs Annalen der Chemie, 1887 , vol. 240, p. 137
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Zincke; Breuer
Justus Liebigs Annalen der Chemie, 1884 , vol. 226, p. 31