反应条件
1: 85 percent / triethylamine / CH2Cl2 / 6 h / 40 °C
2: 85 percent / NaH / dimethylformamide / 1.5 h, RT; 80 deg C, 15 h
3: 93 percent / NaOH / H2O; ethanol / 8 h / 73 °C
View Scheme
参考文献
Kan, Kazunori; Miyama, Akimasa; Hamaguchi, Shigeki; Ohashi, Takehisa; Watanabe, Kiyoshi
Agricultural and Biological Chemistry, 1985 , vol. 49, # 1 p. 207 - 210