D-苯甘氨醇合成路线

参考文献

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620-72-4溴乙酸苯酯+

56613-80-0D-苯甘氨醇

121269-45-2(5R)-3,4,5,6-四氢-5-苯基-4(H)-1,4-恶嗪-2-酮

参考文献

Dellaria, Joseph F.; Santarsiero, Bernard D.
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56613-80-0D-苯甘氨醇

121269-45-2(5R)-3,4,5,6-四氢-5-苯基-4(H)-1,4-恶嗪-2-酮

参考文献

Shafer; Molinski
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2094-74-81-金刚烷甲醛+

56613-80-0D-苯甘氨醇+

151-50-8氰化钾

361441-95-4(alphaS)-alpha-[[(1R)-2-羟基-1-苯基乙基]氨基]-金刚烷-1-乙腈

参考文献

BRISTOL-MYERS SQUIBB COMPANY
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Location in patent: Page/Page column 35 ;
WO 2005/012249 A2

773837-37-9+

2094-74-81-金刚烷甲醛+

56613-80-0D-苯甘氨醇

361441-95-4(alphaS)-alpha-[[(1R)-2-羟基-1-苯基乙基]氨基]-金刚烷-1-乙腈

参考文献

Dong, Jizhe; Gong, Yanchun; Liu, Jun; Chen, Xiangfeng; Wen, Xiaoan; Sun, Hongbin
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56613-80-0D-苯甘氨醇

33911-77-21-[(2R)-2-苯基-1-氮丙啶基]乙酮

参考文献

Ghorai, Manas K.; Shukla, Dipti; Bhattacharyya, Aditya
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75-15-0二硫化碳+

56613-80-0D-苯甘氨醇

110199-18-3(R)-4-苯基噻唑啉-2-硫酮

参考文献

Agami, Claude; Couty, Francois; Prince, Beatrice; Venier, Olivier
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56613-80-0D-苯甘氨醇

110199-18-3(R)-4-苯基噻唑啉-2-硫酮

参考文献

Delaunay, Dominique; Toupet, Loic; Corre, Maurice Le
Journal of Organic Chemistry, 1995 , vol. 60, # 20 p. 6604 - 6607

56613-80-0D-苯甘氨醇

130332-27-33-[[(1R)-2-[[(2R)-2-(2-金刚烷基氧基羰基氨基)-3-(1H-吲哚-3-基)-2-甲基-丙酰]氨基]-1-苯基-乙基]氨基甲酰]丙酸

参考文献

Horwell, David C.; Hughes, John; Hunter, John C.; Pritchard, Martyn C.; Richardson, Reginald S.; at al.
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24424-99-5二碳酸二叔丁酯+

56613-80-0D-苯甘氨醇

67341-01-9N-Boc-DL-苯甘氨醇

参考文献

Skerlj, Renato; Bridger, Gary; Zhou, Yuanxi; Bourque, Elyse; McEachern, Ernest; Metz, Markus; Harwig, Curtis; Li, Tong-Shuang; Yang, Wen; Bogucki, David; Zhu, Yongbao; Langille, Jonathan; Veale, Duane; Ba, Tuya; Bey, Michael; Baird, Ian; Kaller, Alan; Krumpak, Maria; Leitch, David; Satori, Michael; Vocadlo, Krystyna; Guay, Danielle; Nan, Susan; Yee, Helen; Crawford, Jason; Chen, Gang; Wilson, Trevor; Carpenter, Bryon; Gauthier, David; MacFarland, Ron; Mosi, Renee; Bodart, Veronique; Wong, Rebecca; Fricker, Simon; Schols, Dominique
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