反应条件
1: 83 percent / methanol; tetrahydrofuran / 24 h / Ambient temperature
2: 91 percent / H2, aq. NaOH / 10percent Pd/C / methanol / 12 h / 2068.6 Torr / Ambient temperature
3: 84 percent / KOH / H2O / 3 h / Heating
View Scheme
参考文献
Katz; Wise; Townsend
Journal of Medicinal Chemistry, 1982 , vol. 25, # 7 p. 813 - 821