4-(4-吗啉基)苯硼酸频哪醇酯合成路线 （共 3 条）
反应条件
triethylamine; bis-triphenylphosphine-palladium(II) chloride in 1,4-dioxane 4 h; Heating / reflux;
参考文献
SMITHKLINE BEECHAM CORPORATION
Patent: WO2004/13138 A2, 2004 ;
Location in patent: Page 23; 24 ;
WO 2004/013138 A2
反应条件
NiCl2(PMe3)2; TMSOCH2CF3; cesium fluoride in tetrahydrofuran T=100°C; 12 h; Inert atmosphere;
参考文献
Yamamoto, Tetsuya; Morita, Tomoyuki; Takagi, Jun; Yamakawa, Tetsu
Organic Letters, 2011 , vol. 13, # 21 p. 5766 - 5769
反应条件
dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct; potassium acetate in 1,4-dioxane; dichloromethane T=80°C; 12 h;
参考文献
Patel, Gautam; Karver, Caitlin E.; Behera, Ranjan; Guyett, Paul J.; Sullenberger, Catherine; Edwards, Peter; Roncal, Norma E.; Mensa-Wilmot, Kojo; Pollastri, Michael P.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 10 p. 3820 - 3832
