5-溴-4-甲氧基-N,N-二甲基嘧啶-2-胺合成路线 (共 2 条)
反应条件
in tetrahydrofuran
T=20 - 45°C; 0.5 h;
参考文献
Amgen Inc.
Patent: US2006/199817 A1, 2006 ;
Location in patent: Page/Page column 49 ;
US 20060199817 A1
反应条件
n-butyllithium; tri-isopropoxy-borane in tetrahydrofuran; hexane
T=-70 - -20°C; 0.5 h;
参考文献
Amgen Inc.
Patent: US2006/199817 A1, 2006 ;
Location in patent: Page/Page column 49 ;
US 20060199817 A1