1: 4-bromorophenylboronic acid MIDA ester; p-methylphenylboronic acid With potassium phosphate; tetrakis(triphenylphosphine) palladium(0) in 1,4-dioxane T=100°C; 12 h; 2: para-bromoacetophenone in 1,4-dioxane T=100°C; 12 h;
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Location in patent: Page/Page column 23-24 ;
1: With potassium phosphate; Ni(PCy3)2Br2 in tetrahydrofuran T=20°C; Suzuki coupling; Inert atmosphere; 2: With water in tetrahydrofuran T=20°C; Suzuki coupling;
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Xing, Chun-Hui; Lee, Jeng-Ru; Tang, Zhen-Yu; Zheng, Jin Rong; Hu, Qiao-Sheng
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