1-Boc-哌嗪合成路线

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7461-50-94-氨基-2-氯嘧啶+

57260-71-61-Boc-哌嗪

221050-88-01-Boc-4-(2-氯嘧啶-4-基)哌嗪

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WO 2011/095196 A1

3934-20-12,4-二氯嘧啶+

57260-71-61-Boc-哌嗪

221050-88-01-Boc-4-(2-氯嘧啶-4-基)哌嗪+

479691-42-44-(4-氯-嘧啶-2-基)-哌嗪-1-羧酸叔丁酯

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sanofi-aventis
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105-36-2溴乙酸乙酯+

57260-71-61-Boc-哌嗪

209667-59-41-Boc-4-乙氧基羰基甲基哌嗪

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AFFINIUM PHARMACEUTICALS, INC.
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WO 2007/067416 A2

623-73-4重氮乙酸乙酯+

57260-71-61-Boc-哌嗪

209667-59-41-Boc-4-乙氧基羰基甲基哌嗪

参考文献

Varala, Ravi; Enugala, Ramu; Adapa, Srinivas R.
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105-39-5氯乙酸乙酯+

57260-71-61-Boc-哌嗪

209667-59-41-Boc-4-乙氧基羰基甲基哌嗪

参考文献

Meshram; Reddy, B. Chennakesava; Goud, P. Ramesh
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623-48-3碘代醋酸乙酯+

57260-71-61-Boc-哌嗪

209667-59-41-Boc-4-乙氧基羰基甲基哌嗪

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Huang, Wenrong; Naughton, Mary Ann; Yang, Hua; Su, Ting; Dam, Suiko; Wong, Paul W.; Arfsten, Ann; Edwards, Susan; Sinha, Uma; Hollenbach, Stanley; Scarborough, Robert M.; Zhu, Bing-Yan
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57260-71-61-Boc-哌嗪

156478-71-64-Boc-1-哌嗪乙酸

参考文献

WO2013/53983 A1, ;

98-58-8对溴苯磺酰氯+

57260-71-61-Boc-哌嗪

259808-63-4

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F. HOFFMANN-LA ROCHE AG; FIROOZNIA, Fariborz; GILLESPIE, Paul; LIN, Tai-An; MERTZ, Eric; SIDDURI, Achyutharao; SO, Sung-Sau; TAN, Jenny; THAKKAR, Kshitij Chhabilbhai
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WO 2010/055005 A1

506-68-3溴化氰+

57260-71-61-Boc-哌嗪

113534-02-4

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