1-Boc-哌嗪合成路线

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Kuklish, Steven L.; Backer, Ryan T.; Briner, Karin; Doecke, Christopher W.; Husain, Saba; Mullaney, Jeffrey T.; Ornstein, Paul L.; Zgombick, John M.; O'Brien, Thomas P.; Fisher, Matthew J.
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57260-71-61-Boc-哌嗪+

348640-06-24-溴-1H-吡咯并[2,3-b]吡啶

577768-59-34-(1H-吡咯并[2,3-B]吡啶-4-基)-1-哌嗪羧酸叔丁酯

参考文献

GLAXO GROUP LIMITED
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57260-71-61-Boc-哌嗪+

640735-25-74-氟-1-[三(1-甲基乙基)硅酯]-1H-吡咯并[2,3-B]吡啶

577768-59-34-(1H-吡咯并[2,3-B]吡啶-4-基)-1-哌嗪羧酸叔丁酯

参考文献

Caldwell, John J.; Cheung, Kwai-Ming; Collins, Ian
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57260-71-61-Boc-哌嗪

58820-36-31-(4-氯邻甲苯)哌嗪

参考文献

Xiong, Hui; Brugel, Todd A.; Balestra, Michael; Brown, Dean G.; Brush, Kelly A.; Hightower, Caprice; Hinkley, Lindsay; Hoesch, Valerie; Kang, James; Koether, Gerard M.; McCauley Jr., John P.; McLaren, Francis M.; Panko, Laura M.; Simpson, Thomas R.; Smith, Reed W.; Woods, James M.; Brockel, Becky; Chhajlani, Vijay; Gadient, Reto A.; Spear, Nathan; Sygowski, Linda A.; Zhang, Minli; Arora, Jalaj; Breysse, Nathalie; Wilson, Julie M.; Isaac, Methvin; Slassi, Abdelmalik; King, Megan M.
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32315-10-9三光气+

57260-71-61-Boc-哌嗪

59878-28-34-氯羰基-哌嗪-1-羧酸叔丁酯

参考文献

Brinkman, John A.; Cheung, Adrian Wai-Hing; Firooznia, Fariborz; Guertin, Kevin Richard; Marcopulos, Nicholas; Qi, Lida; Racha, Jagdish Kumar; Sarabu, Ramakanth; Tan, Jenny; Tilley, Jefferson Wright
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75-44-5光气+

57260-71-61-Boc-哌嗪

59878-28-34-氯羰基-哌嗪-1-羧酸叔丁酯

参考文献

Rhone-Poulenc Industries
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57260-71-61-Boc-哌嗪+

503-38-8氯甲酸三氯甲酯

59878-28-34-氯羰基-哌嗪-1-羧酸叔丁酯

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Bristol-Myers Squibb Co.
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57260-71-61-Boc-哌嗪

610799-03-64-(氨基磺酰基)哌嗪-1-羧酸叔丁酯

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ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA
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WO 2009/010783 A1

57260-71-61-Boc-哌嗪

622386-08-74-(5-溴吡嗪-2-基)哌嗪-1-羧酸叔丁酯

参考文献

Isabel, Elise; Lachance, Nicolas; Leclerc, Jean-Philippe; Leger, Serge; Oballa, Renata M.; Powell, David; Ramtohul, Yeeman K.; Roy, Patrick; Tranmer, Geoffrey K.; Aspiotis, Renee; Li, Lianhai; Martins, Evelyn
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4701-17-15-溴噻吩-2-甲醛+

57260-71-61-Boc-哌嗪

623588-30-7

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ASTRAZENECA AB
Patent: US2008/153812 A1, 2008 ;
Location in patent: Page/Page column 107 ;
US 20080153812 A1