1: 91 percent / N-ethylmorpholine / CuCl / various solvent(s) / 4 h / 80 °C 2: 10 percent / NaBH4; 2 N aq. NaOH / 48 h / Heating View Scheme
参考文献
Spicer, Julie A.; Gamage, Swarna A.; Rewcastle, Gordon W.; Finlay, Graeme J.; Bridewell, David J. A.; Baguley, Bruce C.; Denny, William A.
Journal of Medicinal Chemistry, 2000 , vol. 43, # 7 p. 1350 - 1358