反应条件
sodium hydride
1.) DMF, 5 min, 2.) DMF, 60 deg C, 30 min; Multistep reaction;
参考文献
Machin, Peter J.; Hurst, David N.; Bradshaw, Rachel M.; Blaber, Leslie C.; Burden, David T.; et al.
Journal of Medicinal Chemistry, 1983 , vol. 26, # 11 p. 1570 - 1576