2-(4-甲氧基苯基)-1H-吲哚合成路线 （共 67 条）
反应条件
1: 55.2 percent / conc. HCl; Sn / ethanol / 6 h / Heating 2: 63.5 percent / m-CPBA / methanol View Scheme
参考文献
Slaett, Johnny; Bergman, Jan
Tetrahedron, 2002 , vol. 58, # 45 p. 9187 - 9191
反应条件
zinc dibromide in toluene
T=130°C; 24 h;
参考文献
Cano, Rafael; Yus, Miguel; Ramon, Diego J.
Tetrahedron, 2012 , vol. 68, # 5 p. 1393 - 1400
反应条件
palladium diacetate; magnesium oxide; triphenylphosphine in 1,4-dioxane; N,N-dimethyl-formamide
T=150°C; 18 h;
参考文献
Sezen, Bengue; Sames, Dalibor
Journal of the American Chemical Society, 2003 , vol. 125, # 18 p. 5274 - 5275
反应条件
PPA
T=70 - 80°C; 0.5 h;
参考文献
Chikvaidze, I. Sh.; Mumladze, E. A.; Samsoniya, Sh. A.; Suvorov, N. N.
Pharmaceutical Chemistry Journal, 1994 , vol. 28, # 10 p. 751 - 755
Khimiko-Farmatsevticheskii Zhurnal, 1994 , vol. 28, # 10 p. 47 - 50
反应条件
dipotassium peroxodisulfate; sulfuric acid in methanol
T=20°C; 10 h;
参考文献
Zhang, Lei; Li, Pinhua; Liu, Can; Yang, Jin; Wang, Min; Wang, Lei
Catalysis Science and Technology, 2014 , vol. 4, # 7 p. 1979 - 1988
反应条件
potassium phosphate; magnesium sulfate; acetic acid; Pd0(tris(tert-butyl)phosphine)2 in N,N-dimethyl acetamide
T=140°C; 21 h;
参考文献
Nazare, Marc; Schneider, Claudia; Lindenschmidt, Andreas; Will, David William
Angewandte Chemie - International Edition, 2004 , vol. 43, # 34 p. 4526 - 4528
反应条件
5 Au/Fe2O3; hydrogen in toluene
T=60 - 120°C; P=750.075 - 15001.5 Torr; 2 h; Autoclave; chemoselective reaction;
参考文献
Yamane, Yoshihiro; Liu, Xiaohao; Hamasaki, Akiyuki; Ishida, Tamao; Haruta, Masatake; Yokoyama, Takushi; Tokunaga, Makoto
Organic Letters, 2009 , vol. 11, # 22 p. 5162 - 5165
反应条件
dicyclohexyl(2′,6′-dimethoxybiphenyl-2-yl)phosphine; palladium diacetate; potassium phosphate in toluene
T=90°C; Suzuki-Miyaura coupling; 2 h;
参考文献
Fang, Yuan-Qing; Lautens, Mark
Journal of Organic Chemistry, 2008 , vol. 73, # 2 p. 538 - 549
反应条件
potassium phosphate; Cu[(phen)(PPh3)2]NO2 in toluene
T=110°C; 6 h;
参考文献
Cacchi, Sandro; Fabrizi, Giancarlo; Parisi, Luca M.
Organic Letters, 2003 , vol. 5, # 21 p. 3843 - 3846
反应条件
copper(l) iodide; potassium carbonate; L-proline in N,N-dimethyl-formamide
T=80°C; 24 h;
参考文献
Liu, Feng; Ma, Dawei
Journal of Organic Chemistry, 2007 , vol. 72, # 13 p. 4844 - 4850
