(2-氨基-4-氟苯基)-氨基甲酸-1,1-二甲基乙酯合成路线 (共 2 条)
反应条件
sodium dithionite; water; sodium hydrogencarbonate in tetrahydrofuran; methanol T=20°C; 0.5 h;
参考文献
PHARMACOPEIA , INC.
Patent: WO2008/60301 A1, 2008 ;
Location in patent: Page/Page column 63-64 ;
反应条件
in tetrahydrofuran T=20°C; 6 h;
参考文献
CURIS, INC.; QIAN, Changgeng; CAI, Xiong; ZHAI, Haixiao
Patent: WO2010/75542 A1, 2010 ;
Location in patent: Page/Page column 78 ;