反应条件
1: 90.3 percent / imidazole / dimethylformamide / 20 h / Ambient temperature 2: 31.58 percent / MoOPH, lithium diisopropylamide / hexane; tetrahydrofuran / 1.5 h / -44 °C 3: 95.15 percent / 30percent aq. HF / acetonitrile / 1.5 h / Ambient temperature View Scheme
参考文献
Geier, Martina; Braun, Andreas; Fladischer, Patrik; Stepniak, Piotr; Rudroff, Florian; Hametner, Christian; Mihovilovic, Marko D.; Glieder, Anton
FEBS Journal, 2013 , vol. 280, # 13 p. 3094 - 3108