反应条件
1: 1.) aq. NaOH / 1.) EtOH, reflux, 25 min, 2.) DMF, 60 deg C, 24 h 2: NaBH4 / methanol; diethyl ether View Scheme
参考文献
Cavallaro, Rosaria A.; Filocamo, Luigi; Galuppi, Annamaria; Galione, Antony; Brufani, Mario; Genazzani, Armando A.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 14 p. 2527 - 2534