反应条件
1: [3H]-Indoleacetic acid With HATU in N,N-dimethyl-formamide
T=20°C; 0.5 h;
2: 1-methyl-piperazine in N,N-dimethyl-formamide
4 h;
参考文献
MYREXIS, INC.; KUMAR, Dange Vijay; SLATTUM, Paul M.; YAGER, Kraig M.; SHENDEROVICH, Mark D.; TANGALLAPALLY, Rajendra; KIM, Se-Ho
Patent: WO2012/177782 A1, 2012 ;
Location in patent: Page/Page column 99-100 ;
WO 2012/177782 A1
