反应条件
1: 74 percent / DMAP, 2,6-lutidine / CH2Cl2; tetrahydrofuran / -78 - 0 °C 2: 84 percent / Pd(OAc)2, dppp, Et3N / dimethylsulfoxide / 5 h / 70 °C View Scheme
参考文献
Yao, Zhu-Jun; Ye, Bin; Wu, Xiong-Wu; Wang, Shaomeng; Wu, Li; Zhang, Zhong-Yin; Burke Jr., Terrence R.
Bioorganic and Medicinal Chemistry, 1998 , vol. 6, # 10 p. 1799 - 1810