反应条件
potassium phosphate; palladium diacetate; 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene; sodium t-butanolate in toluene
T=140°C; 24 h; Molecular sieve;
参考文献
BLEND THERAPEUTICS; BILODEAU, Mark, T.; DUNBAR, Craig, A.; BARDER, Timothy, E.; LEE, Edward, R.; ALARGOVA, Rossitza, G.; ROCKWOOD, Danielle, N.; MOREAU, Benoit; SHINDE, Rajesh; BOUTHILLETTE, Melaney
Patent: WO2014/43243 A2, 2014 ;
Location in patent: Paragraph 00249 ;