反应条件
1: 100 percent / imidazole, DMAP / dimethylformamide / 10 h / Ambient temperature 2: 97 percent / Me3Al / CH2Cl2; hexane / 1.) -15 deg C, 30 min; room temp., 35 min, 2.) room temp., 2 h View Scheme
参考文献
Ascenso, Osvaldo S.; Marques, Joao C.; Santos, Ana Rita; Xavier, Karina B.; Rita Ventura; Maycock, Christopher D.
Bioorganic and Medicinal Chemistry, 2011 , vol. 19, # 3 p. 1236 - 1241