反应条件
1: 80 percent / CH2Cl2 / Ambient temperature
2: 1.) POCl3, DMF, 2.) DMF, Et3N / 1.) CH2Cl2, reflux, 14 h, 2.) CH2Cl2, 0 deg C to rt
View Scheme
参考文献
Ghosez, Leon; George-Koch, Isabelle; Patiny, Luc; Houtekie, Marc; Bovy, Philippe; Nshimyumukiza, Prosper; Phan, Thao
Tetrahedron, 1998 , vol. 54, # 31 p. 9207 - 9222