反应条件
1: With 4-(N,N-dimethlyamino)pyridine; N'-(3-dimethylaminopropyl)-N-ethylcarbodiimide in N,N-dimethyl-formamide T=25°C; 4 h; 2: With sodium hydroxide in N,N-dimethyl-formamide T=100°C; 10 h;
参考文献
He, Yun; Yang, Jun; Wu, Baogen; Robinson, Dale; Sprankle, Kelly; Kung, Pei-Pei; Lowery, Kristin; Mohan; Hofstadler, Steve; Swayze, Eric E.; Griffey, Rich
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 3 p. 695 - 699