1: tetrakis(triphenylphosphine) palladium(0); potassium carbonate / tetrahydrofuran; water / 80 °C / |Inert atmosphere
2: toluene-4-sulfonic acid; sodium nitrite; potassium iodide / water; acetonitrile / 4 h / 10 - 20 °C
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参考文献
Tran-Van, Anne-Florence; Huxol, Elena; Basler, Jonathan M.; Neuburger, Markus; Adjizian, Jean-Joseph; Ewels, Chris P.; Wegner, Hermann A.
Organic Letters, 2014 , vol. 16, # 6 p. 1594 - 1597
Blackaby, Wesley Peter; Goodacre, Simon Charles; Hallett, David James; Jennings, Andrew; Lewis, Richard Thomas; Moore, Kevin William; Street, Leslie Joseph
Patent: US2003/176449 A1, 2003 ;