间溴苯酚合成路线

591-20-8间溴苯酚

207122-16-52,2’,3,4,4’,5,6-七溴联苯醚

参考文献

Liu, Huiling; Bernhardsen, Monica; Fiksdahl, Anne
Tetrahedron, 2006 , vol. 62, # 15 p. 3564 - 3572

110-91-8吗啉+

591-20-8间溴苯酚

27292-49-53-(4-吗啉基)苯酚

参考文献

Advanced Synthesis and Catalysis, , vol. 346, # 6 p. 611 - 616

591-20-8间溴苯酚+

141699-59-41-Boc-4-甲烷磺酰氧基哌啶

790667-54-81-BOC-4-(3-溴苯氧基)哌啶

参考文献

AURIGENE DISCOVERY TECHNOLOGIES LIMITED; UM PHARMAUJI SDN. BHD; GUMMADI, Venkateshwar, Rao; HOSAHALLI, Subramanya; NANDURI, Srinivas; AGGUNDA RENUKAPPA, Girish
Patent: WO2014/6554 A1, 2014 ;
Location in patent: Page/Page column 43; 44 ;

591-20-8间溴苯酚+

118811-07-74-(甲苯-4-磺酰氧)哌啶-1-羧酸叔丁酯

790667-54-81-BOC-4-(3-溴苯氧基)哌啶

参考文献

Sato, Kenjiro; Sugimoto, Hiromichi; Rikimaru, Kentaro; Imoto, Hiroshi; Kamaura, Masahiro; Negoro, Nobuyuki; Tsujihata, Yoshiyuki; Miyashita, Hirohisa; Odani, Tomoyuki; Murata, Toshiki
Bioorganic and Medicinal Chemistry, 2014 , vol. 22, # 5 p. 1649 - 1666

591-20-8间溴苯酚+

109384-19-2N-Boc-4-羟基哌啶

790667-54-81-BOC-4-(3-溴苯氧基)哌啶

参考文献

KADMON CORPORATION, LLC; BOXER, Michael; RYAN, John; TONRA, James
Patent: WO2014/55999 A2, 2014 ;
Location in patent: Paragraph 0238 ;

591-20-8间溴苯酚

855836-52-12-碘-3-溴苯酚

参考文献

Sanz, Roberto; Castroviejo, M. Pilar; Fernandez, Yolanda; Fananas, Francisco J.
Journal of Organic Chemistry, 2005 , vol. 70, # 16 p. 6548 - 6551

591-20-8间溴苯酚

30724-22-23-(三氟甲氧基)苯乙酮

参考文献

Blencowe, Anton; Cosstick, Kevin; Hayes, Wayne
New Journal of Chemistry, 2006 , vol. 30, # 1 p. 53 - 58

591-20-8间溴苯酚+

108-24-7乙酸酐

30186-18-64-溴-2-羟基苯乙酮

参考文献

DAC S.r.l.
Patent: EP2110377 A1, 2009 ;
Location in patent: Page/Page column 15 ;

591-20-8间溴苯酚+

75-36-5乙酰氯

30186-18-64-溴-2-羟基苯乙酮

参考文献

Takeda Pharmaceutical Company Limited
Patent: EP1921066 A1, 2008 ;
Location in patent: Page/Page column 70 ;

89368-12-74-溴-2-甲氧基苯乙酮

30186-18-64-溴-2-羟基苯乙酮+

35065-86-23-溴乙酸苯酯

参考文献

US5332757 A1, ;
US 5332757 A